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Eletriptan hydrobromide
CAS No. 177834-92-3
Eletriptan hydrobromide ( UK 116044 hydrobromide )
产品货号. M12677 CAS No. 177834-92-3
Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥267 | 有现货 |
|
| 5MG | ￥421 | 有现货 |
|
| 10MG | ￥518 | 有现货 |
|
| 25MG | ￥1102 | 有现货 |
|
| 50MG | ￥2001 | 有现货 |
|
| 100MG | ￥3645 | 有现货 |
|
| 200MG | ￥4739 | 有现货 |
|
| 500MG | ￥7590 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Eletriptan hydrobromide
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist.
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产品描述Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist; significantly increases occluded wedge pressure and mean pulmonary artery pressure in vivo, with no significant coronary artery constriction, and obstructive coronary artery disease; displays antimigraine activity.Migrainev Approved
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同义词UK 116044 hydrobromide
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体5-HT1B;5-HT1D
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研究领域Neurological Disease
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适应症Migraine
化学信息
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CAS Number177834-92-3
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分子量463.43
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分子式C22H26N2O2S.HBr
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纯度>98% (HPLC)
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溶解度DMSO: 46.3 mg/mL (100 mM) （ < 1 mg/ml refers to the product slightly soluble or insoluble )
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SMILESCN1CCC[C@@H]1CC2=CNC3=C2C=C(C=C3)CCS(=O)(=O)C4=CC=CC=C4.Br
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化学全称3-[[(2R)-1-Methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-indole hydrobromide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Napier C, et al. Eur J Pharmacol. 1999 Mar 5;368(2-3):259-68.
2. Gupta P, et al. Eur J Pharmacol. 1999 Feb 19;367(2-3):283-90.
3. Muir DF, et al. Clin Pharmacol Ther. 1999 Jul;66(1):85-90.
2. Gupta P, et al. Eur J Pharmacol. 1999 Feb 19;367(2-3):283-90.
3. Muir DF, et al. Clin Pharmacol Ther. 1999 Jul;66(1):85-90.
产品手册
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